Inhibitor (μM) | Cell line | Two-dimensional | Three-dimensional |
---|---|---|---|
17-AAG: | U-87 MG | 0.43 ± 0.13 | 0.82 ± 0.16 |
 | KNS42 | 18.02 ± 6.42 | 81.43 ± 1.60 |
 | MDA-MB-231 P | 2.47 ± 0.83 | 2.33 ± 0.33 |
 | MDA-MB-231 M | 0.75 ± 0.10 | 6.19 ± 0.50 |
 | LICR-LON-HN4 | 0.07 ± 0.06 | 0.38 ± 0.11 |
PI-103: | U-87 MG | 0.49 ± 0.13 | 0.16 ± 0.03 |
 | KNS42 | 2.15 ± 1.20 | 0.72 ± 0.34 |
 | MDA-MB-231 P | 2.39 ± 0.69 | > 100 |
CCT130234: | U-87 MG | 9.10 ± 1.13 | 16.40 ± 0.14 |
 | MDA-MB-231 P | 11.5 ± 3.32 | 8.50 ± 0.62 |