From: Targeting the Tie2–αvβ3 integrin axis with bi-specific reagents for the inhibition of angiogenesis
Integrin | KD ± sem, nM | Kon1 ± sem (M−1 s−1) × 104 | Koff1 ± sem (s−1) × 10−3 | Kon2 ± sem (s−1) × 10−3 | Koff2 ± sem (s−1) × 10−3 |
---|---|---|---|---|---|
αvβ1 | 550 ± 90.1 | 1.14 ± 0.01 | 6.29 ± 0.17 | 3.04 ± 0.12 | 1.97 ± 0.03 |
αvβ5 | 65 ± 21.8 | 3.98 ± 0.03 | 2.59 ± 0.12 | 5.44 ± 0.21 | 0.35 ± 0.01 |
αvβ6 | 364 ± 70.8 | 2.29 ± 0.05 | 8.35 ± 0.45 | 3.2 ± 0.17 | 1.06 ± 0.03 |
αvβ8 | 138 ± 50.3 | 3.66 ± 0.03 | 5.05 ± 0.13 | 2.4 ± 0.12 | 2.15 ± 0.05 |